|
|
科研情况: |
|
近年来主持国家自然基金青年项目、陕西省教育厅创新团队项目、三秦英才计划区域人才项目以及咸阳市科技局项目;参与2项国家自然基金面上项目。 1. 陕西省教育厅,创新团队项目,22JP019,基于秦皮活性物质香豆素的衍生物合成和抗肿瘤活性研究,2022-2023,5万元,主持; 2. 国家自然科学基金委员会,青年基金项目,82204235,色胺酮治疗溃疡性结肠炎的代谢研究和靶向前药设计合成,2023-2025,30万元,主持; 3. 陕西省组织部,三秦英才计划-人才引进区域人才项目,青黛治疗溃疡性结肠炎活性和物质基础研究,2024-2026,30万。 4. 咸阳市科技局,L2024-Q CY-ZYYJJQ-X193,色胺酮衍生物合成和抗溃疡性结肠炎研究,2024-2025,5万元,主持。 5. 咸阳市创新能力支撑计划-科技创新人才(教育科技人才一体化)专项,青黛抗溃疡性结肠炎的机制研究以及基于活性成分的创新药物研制,L2025-CXNL-KJRC-004,2025.-2027,2万,主持。 |
|
代表性论文: |
|
1. Mao-Hao Li, Zheng Wang, Yanni Liang, Simeng Lu, Bao-Long Hou*. Synthesis, characterization, crystal structure, and anti-inflammatory evaluation of thienyl-substituted tryptanthrins, J. Mol. Stru., 2025, 1342, 142651. 2. Bao-Long Hou, Wenyu Li, Ruirui Feng, Xiumei Yang, Jianli Liu, Cuiling Wang*. A novel rhodamine 6G-based chemosensor for Fe3+ detection in water samples and cellular imaging, Results in Chem., 2025,15, 102228。 3. 侯宝龙*,李茂浩.地椒草精油体外抗炎和抗氧化活性研究.天然产物研究与开发, 2025,37(09):1679-1688. 4. Bao-Long Hou, Kenan Wu, Rongrong Liu, et al. Natural products fragment-based design and synthesis of a novel pentacyclic ring system as potential MAPK inhibitor, Bioorg. Med. Chem. Lett., 2024, 99,129598. 5. Bao-Long Hou, Junyang Liu, Chuang Qiao, Chuang-Chuang Li. Total synthesis of natural products containing bicyclo[n.2.2] ring systems, Tetrahedron Lett., 2024, 135, 154871. 6. Bao-Long Hou, Jiaxu Yan, Rongrong Liu, et al. Bcr-Abl inhibitory activities of imatinib derivatives, Lett. Drug. Design. Discov., 2024, 21, 4085. 7. Cuiling Wang, Ying Zhou, RongRong Liu,....Bao‑Long Hou*. A novel tryptanthrin-based “on–off-on” probe for sequential sensing Cu2+/S2− in water samples, Anal. Sci., 2024, 40, 1279. 8.侯宝龙,李雯钰,尚东院,刘建利,王翠玲.色胺酮衍生物的设计合成及其抗肿瘤和抗菌活性研究,中国药物化学杂志,2023, 33, 820. 9. He, Y. T.; Li, L-X.; Lin, X. H.; Bao-Long Hou; Li, C.-C*. Synthesis of Various Bridged Ring Systems via Rhodium-Catalyzed Bridged (3+2) Cycloadditions. Org. Lett. 2022, 24, 186–190. 10. Bao-Long Hou; Wong, J. J.; Lv, N.; Wang, Y. Q.; Houk, K. N.; Li, C. -C*. Facile Generation of Bridged Medium-sized Polycyclic Systems by Type II Intramolecular (3+2) Dipolar Cycloadditions. Nat. Commu. 2021, 12, 5239. Bao-Long Hou; Li, L.-X.; Li, C.-C*. Synthesis of the Bridged [5-7-7] Tricyclic Core of Eurifoloid A. Org. Lett. 2021,23, 7771-7775. 11. Bao-Long Hou,; Zhou, Y; Li, W. Y.; Liu, J. L; Wang, C. L*. Synthesis and Evaluation of Tryptanthrins as Antitumor Agents. Tetrahedron 2021, 99, 132454. 12. 侯宝龙,王征,梁艳妮。一种色胺酮类化合物及其制备方法与应用,专利号:ZL20251 0609256.0 |
|
荣誉奖励: |
|
三秦英才计划区域人才项目(2024) 咸阳市科技创新人才(2025) |
|
工作经历: |
|
2016-2018 南方科技大学-华南理工大学 博士后 2018-2021 南方科技大学 高级研究学者
|
|
地址:陕西省西咸新区世纪大道 邮编:712046 电话:029-38185000
版权所有:陕西中医药大学 技术支持:信息化建设管理处 陕ICP备05001612号-1
陕公网安备 61040202000395号